产品详情
简单介绍：
CAS:1255580-76-7Formula:C30H47N5O2MW:509.72Appearance:Off-whitesolidPurity:≥98%byHPLC
详情介绍：
Cell-permeable. UNC0638 is a potent G9a HMTase inhibitor, exhibiting an IC50 value of 50 value of 19 nM, but is more than 10,000-fold selective against SET7/9 (a H3K4 HMTase), SET8 (a H4K20 HMTase), PRMT3, and SUV39H2. UNC0638 inhibits H3K9 dimethylation in MDA-MB231 cells with an IC50 value of 81 nM and demonstrates favorable separation of functional and toxic effect.
Additional Information
| Product # | U-2473 |
|---|---|
| CAS # | 1255580-76-7 |
| Chemical Name | 2-Cyclohexyl-6-methoxy-N-[1-(1-methylethyl)-4-piperidinyl]-7-[3-(1-pyrrolidinyl)propoxy]-4-quinazolinamine |
| Formula | C30H47N5O2 |
| MW | 509.72 |
| Appearance | Off-white solid |
| Purity | ≥98% by HPLC |
| Solubility | DMSO (10 mM) |
| Storage Temp | -20°C |
Additional Information
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