XAV-939; XAV-939;284028-89-3
Formula:C14H11F3N2OS
Molecular Weight:312.31
Appearance:White to off-white powder
Purity:98+%
XAV-939 (NVP-XAV939) selectively inhibits Wnt/β-catenin-mediated transcription through tankyrase1/2 inhibition with IC50 of 11 nM/4 nM in cell-free assays, regulates axin levels and does not affect CRE, NF-κB or TGF-β.